Bildiriler
- A STUDY ABOUT ANTIPROLIFERATIVE EFFECT OF A4B3 ON HUMAN LUNG CANCER CELLS (A549)26.06.2018 - 26.06.2018Özet bildiriUluslararasıİngilizce12th International Symposium on Pharmaceutical SciencesAYDIN HASAN, YUMRUTAŞ ÖNDER, LOLAK NEBİH, AKOCAK SÜLEYMANIn Silico Studies and Antibacterial Evaluation of N,n`-Diaryl Cyanoguanidine-Substituted Sulfonamides28.08.2021 - 28.08.2021Özet bildiriUluslararasıİngilizce7th International Medicine and Health Sciences Researches CongressLOLAK NEBİH, AKOCAK SÜLEYMANhttp://www.utsakcongress.com/prog-ve-ozet-kitap.htmlYeni Sülfisoksazol ve Sülfaguanidin türevi bis-ürelerin sentezi ve bu moleküllerinçeşitli metabolic enzimlere karşı enzim inhibisyon çalışmaları22.08.2020 - 22.08.2020Özet bildiriUluslararasıİngilizce4 th International Medicine and Health Sciences Researches Congress( UTSAK )LOLAK NEBİHSynthesis and Properties of Novel Hydroxylamino-Substituted 1,2,4–Oxadiazoles and 1,2,4–Triazole17.06.2008 - 17.06.2008Özet bildiriUluslararasıİngilizceThe Fifth Jordanian International Conference of ChemistryGeffken Detlef,LOLAK NEBİHhttp://chem.yu.edu.jo/conf/index.htmYeni sülfonamit içerem N,N`-arilsiyanoguanidinlerin sentezi ve karbonik anhidraz izoenzimleri hCA I, II, IV ve IX üzerine inhibisyon testleri.22.03.2018 - 22.03.2018Özet bildiriUlusalTürkçeUluslararası Katılımlı 6. İlaç Kimyası: İlaç Etkin Maddesi Tasarımı, Sentezi, Üretimi ve Standardizasyonu Kongresi.LOLAK NEBİH,AKOCAK SÜLEYMAN,BUA Silvia,SUPURAN Claudiu TYeni histamine Schiff bazı türevlerinin sentezi ve çeşitli karbonik anhidraz izoenzimleri üzerine aktivasyon testleri22.03.2018 - 22.03.2018Özet bildiriUlusalTürkçeUluslararası Katılımlı 6. İlaç Kimyası: İlaç Etkin Maddesi Tasarımı, Sentezi, Üretimi ve Standardizasyonu Kongresi.AKOCAK SÜLEYMAN,LOLAK NEBİH,DURGUN MUSTAFA,VULLO Daniela,SUPURAN Claudiu TYeni 1,3-triazen türevi metanilamit ve sülfonilamitlerin sentezi ve karbonik anhidraz izoenzimleri hCA I, II, VII ve IX üzerine inhibisyon testleri.22.03.2018 - 22.03.2018Özet bildiriUlusalTürkçeUluslararası Katılımlı 6. İlaç Kimyası: İlaç Etkin Maddesi Tasarımı, Sentezi, Üretimi ve Standardizasyonu KongresiAKOCAK SÜLEYMAN,LOLAK NEBİH,TUNEG Muhammed,SUPURAN Claudiu THistamin Schiff Bazı Türevlerinin Sentezi, Antioksidan ve Antikolinesteraz Aktivitelerinin Araştırılması14.03.2019 - 14.03.2019Özet bildiriUluslararasıİngilizce7th Drug Chemistry Conference:Design, Synthesis, Production and Standardization of Drug Active SubstancesAKOCAK SÜLEYMAN,LOLAK NEBİH,TUNEG Muhammed,BOĞA MEHMETSpinaceamin türevi bileşiklerin çeşitli α-karbonik anhidraz izoenzimleri üzerine aktivasyon testleri.14.03.2019 - 14.03.2019Özet bildiriUluslararasıİngilizce7th Drug Chemistry Conference:Design, Synthesis, Production and Standardization of Drug Active SubstancesAKOCAK SÜLEYMAN,LOLAK NEBİH,BUA Silvia,KARAKOÇ Gülçin,SUPURAN Claudiu TYeni 1,3,5-triazin içeren benzensülfonamitlerin sentez edilmesi ve karbonik anhidraz izoenzimleri hCA I, II, IX ve XII üzerine inhibisyon testleri14.03.2019 - 14.03.2019Özet bildiriUluslararasıİngilizce7th Drug Chemistry Conference:Design, Synthesis, Production and Standardization of Drug Active SubstancesLOLAK NEBİH,AKOCAK SÜLEYMAN,BUA Silvia,SUPURAN Claudiu T1,3-diariltriazen sübstittüe sülfonamitlerin sentezi, antioksidan ve antikolinesteraz aktivitelerinin araştırılması.14.03.2019 - 14.03.2019Özet bildiriUluslararasıİngilizce7th Drug Chemistry Conference:Design, Synthesis, Production and Standardization of Drug Active SubstancesAKOCAK SÜLEYMAN,LOLAK NEBİH,BOĞA MEHMET,TUNEG MuhammedKarbonik anhidraz içeren kanser türlerini inhibe eden Bis yapılı sülfonamitlerin sentezi ve bu bileşiklerin biyolojik testleri30.03.2017 - 30.03.2017Özet bildiriUlusalTürkçe5. İlaç Kimyası: İlaç Etkin Maddesi Tasarımı, Sentezi, Üretimi ve Standardizasyonu KongresiAKOCAK SÜLEYMAN,LOLAK NEBİH,DURGUN MUSTAFA,SUPURAN Claudiu T,İLİES Marc APotent and Selective Inhibition of Carbonic Anhydrase Isoforms by Using 1,3,5-triazine and 1,3-diaryltriazene Substituted Sulfonamides27.02.2020 - 27.02.2020Özet bildiriUluslararasıİngilizce8th International of Drug Chemistry CoferenceAKOCAK SÜLEYMAN,LOLAK NEBİH,Claudiu T SUPURANhttps://ilackongresi.org/wp-content/uploads/8-ilac-kongresi-kitapcik_compressed.pdfAromatik Yapıya Sahip Bis-Sülfonamit Schiff Bazı Türevlerinin Sentezi, Antioksidan, Asetilkolinesteraz ve Bütirilkolinesteraz Aktivitelerinin Araştırılması27.02.2020 - 27.02.2020Özet bildiriUluslararasıİngilizce8th International of Drug Chemistry CoferenceTUNEG Muhammed,LOLAK NEBİH,BOĞA MEHMET,AKOCAK SÜLEYMANhttps://ilackongresi.org/wp-content/uploads/8-ilac-kongresi-kitapcik_compressed.pdf1,3,5-Triazin Türevi Üreido Benzen Sülfonamitlerin Sentezi, Antioksidan, Asetilkolinesteraz, Bütirilkolinesteraz ve Tirozinaz Enzim Aktivitelerinin Araştırılması27.02.2020 - 27.02.2020Özet bildiriUluslararasıİngilizce8th International Drug Chemistry ConferenceLOLAK NEBİHhttps://ilackongresi.org/wp-content/uploads/8-ilac-kongresi-kitapcik_compressed.pdfSynthesize of new histamine Schiff base derivatives as an isoform-selective and potent carbonic anhydrase VII activators27.06.2018 - 27.06.2018Özet bildiriUluslararasıİngilizce11th International Conference on Carbonic Anhydrases,AKOCAK SÜLEYMAN,LOLAK NEBİH,VULLO Daniela,DURGUN MUSTAFA,SUPURAN Claudiu TEvaluation of Anti-proliferative effect of novel synthesized 4-(3-(4-fluorophenyl)triaz-1-en-1-yl) benzenesulfonamide on Lung cancer cell line (A549)11.10.2017 - 11.10.2017Özet bildiriUluslararasıİngilizce2nd International Gazi Pharma Symposium SeriesAYDIN HASAN,AKOCAK SÜLEYMAN,LOLAK NEBİH,YUMRUTAS Onder1,3-Triazen türevi benzen sülfonamitlerin sentezi kanserle ilgili karbonik anhidraz izoenzimlerini inhibe etme özelliklerinin testi.30.03.2017 - 30.03.2017Özet bildiriUlusalTürkçe5. İlaç Kimyası: İlaç Etkin Maddesi Tasarımı, Sentezi, Üretimi ve Standardizasyonu KongresiLOLAK NEBİH,AKOCAK SÜLEYMAN,TEKELİ YENER,SUPURAN Claudiu TSynthesis and biological evaluation of aromatic and heterocyclic Bis-sulfonamide Schiff bases as carbonic anhydrase I, II, VII, and IX inhibitors24.05.2017 - 24.05.2017Özet bildiriUluslararasıİngilizce3rd Satellite Meeting on Carbonic Anhydrase, Montecatini TermeAKOCAK SÜLEYMAN,LOLAK NEBİH,NOCENTİNİ Alessio,TEKELİ YENER,SUPURAN Claudiu TAromatik ve heterosiklik Bis yapılı sülfonamitlerin sentezi ve kanserle ilgili karbonik anhidraz izoenzimleri üzerine inhibisyon testleri30.03.2017 - 30.03.2017Özet bildiriUlusalTürkçe5. İlaç Kimyası: İlaç Etkin Maddesi Tasarımı, Sentezi, Üretimi ve Standardizasyonu KongresiAKOCAK SÜLEYMAN,LOLAK NEBİH,KARAKOÇ Gülçin,TUFAN Anzel,SUPURAN Claudiu TSynthesis of 1,3-Triazene substituted benzenesulfoanmides and testing their carbonic anhydrase inhibition properties against I, II, VII, and IX isozymes24.05.2017 - 24.05.2017Özet bildiriUluslararasıİngilizce3rd Satellite Meeting on Carbonic Anhydrase, Montecatini TermeAKOCAK SÜLEYMAN,TEKELİ YENER,BUA Silvia,LOLAK NEBİH,SUPURAN Claudiu T
Makaleler
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Medicinal Chemistry Letters0960-894XAKOCAK SÜLEYMAN, LOLAK NEBİH, Giovannuzzi Simone, Supuran Claudiu Thttp://dx.doi.org/10.1016/j.bmcl.2023.129479Evaluation of cytotoxic, antifungal, and larvicidal activities of different bis‐sulfonamide Schiff base compounds5.2023HakemliÖzgün MakaleUluslararasıİngilizceJournal of Biochemical and Molecular Toxicology1095-6670AYDIN HASAN, AKOCAK SÜLEYMAN, LOLAK NEBİH, YUMRUTAŞ ÖNDER, USLU UĞUR, BOZGEYİK İBRAHİM, ÜÇKARDEŞ FATİH, GÜNAL SELAMİ, CEYLAN ONURhttp://dx.doi.org/10.1002/jbt.23375Design and Synthesis of Pyrazole Carboxamide Derivatives as Selective Cholinesterase and Carbonic Anhydrase Inhibitors: Molecular Docking and Biological Evaluation1.2023HakemliÖzgün MakaleUluslararasıTürkçeWiley1612-1872DURGUN MUSTAFA, AKOCAK SÜLEYMAN, LOLAK NEBİH, TOPAL FEVZİ, KOÇYİĞİT ÜMİT MUHAMMET, TÜRKEŞ CÜNEYT, IŞIK MESUT, BEYDEMİR ŞÜKRÜhttp://dx.doi.org/10.1002/cbdv.202301824Potent carbonic anhydrase I, II, IX and XII inhibition activity of novel primary benzenesulfonamides incorporating bis-ureido moieties3.2023HakemliÖzgün MakaleUluslararasıİngilizceJournal of Enzyme Inhibition and Medicinal Chemistry1475-6374TEKELİ TUBA, AKOCAK SÜLEYMAN, Petreni Andrea, LOLAK NEBİH, ÇETE SERVET, Supuran Claudiu T.https://www.tandfonline.com/doi/full/10.1080/14756366.2023.2185762Antibacterial, Antioxidant and DNA Cleavage Activity Evaluation of Substituted Phenylureido Sulfaguanidine and Sulfamethazine Derivatives6.2022HakemliÖzgün MakaleUluslararasıİngilizcePharmaceutical Chemistry Journal0023-1134TEKELİ YENER, LOLAK NEBİH, DENİZ SÖNMEZ GÖRKEM, TEKELİ TUBA, AKOCAK SÜLEYMANhttps://link.springer.com/content/pdf/10.1007/s11094-022-02654-7.pdfBiological evaluation of aromatic bis-sulfonamide Schiff bases as antioxidant, acetylcholinesterase and butyrylcholinesterase inhibitors6.2020HakemliÖzgün MakaleUlusalİngilizceCumhuriyet University2587-2680LOLAK NEBİH,AKOCAK SÜLEYMANhttp://dx.doi.org/10.17776/csj.595463Novel inhibitors with sulfamethazine backbone: 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Journal0091-150XLOLAK NEBİH, BOĞA MEHMET, DENİZ SÖNMEZ GÖRKEM, Tuneğ Muhammed, DOĞAN ASLINUR, AKOCAK SÜLEYMANhttp://dx.doi.org/10.1007/s11094-022-02581-7In Silico Molecular Docking Study on Selective Cyclooxygenase-2 Inhibitor Drugs For SARS-Cov-2 Active Main Protease1.2022HakemliÖzgün MakaleUluslararasıİngilizceNovel Approaches in Drug Designing & Development2575-8942DOĞAN ASLINUR, ŞENGÜL FATMA, LOLAK NEBİH, AKOCAK SÜLEYMANhttps://juniperpublishers.com/napdd/articleinpress-napdd.phpBimetallic PdRu/graphene oxide based Catalysts for one-pot three-component synthesis of 2-amino-4H-chromene derivatives10.2017HakemliÖzgün MakaleUluslararasıİngilizceNano-Structures Nano-Objects2352-507XŞEN BETÜL,LOLAK NEBİH,PARALI ÖZGE,KOCA MURAT,Şavk Aysun,AKOCAK SÜLEYMAN,ŞEN FATİHhttps://linkinghub.elsevier.com/retrieve/pii/S2352507X17301610Synthesis and biological evaluation of 1,3,5-triazine-substituted ureido benzenesulfonamides as antioxidant, acetylcholinesterase and butyrylcholinesterase 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Thttps://www.tandfonline.com/doi/full/10.1080/14756366.2018.1515933Synthesis and biological evaluation of novel N,N′-diaryl cyanoguanidines acting as potent and selective carbonic anhydrase II inhibitors4.2018HakemliÖzgün MakaleUluslararasıİngilizceBIOORGANIC CHEMISTRY0045-2068AKOCAK SÜLEYMAN,LOLAK NEBİH,Bua Silvia,Turel Idris,Supuran Claudiu Thttps://linkinghub.elsevier.com/retrieve/pii/S0045206817309331Synthesis and biological evaluation of histamine Schiff bases as carbonic anhydrase I, II, IV, VII, and IX activators1.2017HakemliÖzgün MakaleUluslararasıİngilizceJOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY1475-6366AKOCAK SÜLEYMAN,LOLAK NEBİH,Vullo Daniela,DURGUN MUSTAFA,Supuran Claudiu Thttps://www.tandfonline.com/doi/full/10.1080/14756366.2017.1386660Biological effects of a new set 1,2,4-triazolo[1,5-a]quinazolines on heart rate and blood pressure12.2014HakemliÖzgün MakaleUluslararasıİngilizceChemistry Central Journal1752-153XAl-Salahi Rashad,El-Tahir Kamal-Eldin,Alswaidan Ibrahim,LOLAK NEBİH,Hamidaddin Mohammed,Marzouk Mohamedhttps://bmcchem.biomedcentral.com/articles/10.1186/1752-153X-8-3Rapid and efficient microwave-assisted synthesis of 5-amino-3-aralkoxy(methoxy)amino-1,2,4-oxadiazoles4.2007HakemliÖzgün MakaleUluslararasıİngilizceTETRAHEDRON LETTERS0040-4039Kurz Thomas,LOLAK NEBİH,Geffken Detlefhttps://linkinghub.elsevier.com/retrieve/pii/S0040403907003358Correction to “Composites of Palladium−Nickel Alloy Nanoparticles and Graphene Oxide for the Knoevenagel Condensation of Aldehydes with Malononitrile”10.2020HakemliTeknik NotUluslararasıİngilizceACS Omega2470-1343","2470-1343LOLAK NEBİH, Kuyuldar Esra, BURHAN Hakan, GÖKSU HAYDAR, AKOCAK SÜLEYMAN, ŞEN FATİHhttps://pubs.acs.org/doi/pdf/10.1021/acsomega.0c043832-Phenoxy-1,2,4-triazolo[1,5-a]quinazolin-5(4H)-one.6.2012HakemliÖzgün MakaleUluslararasıİngilizceActa Crystallographica Section E Structure Reports Online1600-5368Al-Salahi Rashad,LOLAK NEBİH,Al-Omar Mohamed,Ng Seik Weng